Neuroprotective Effect of a New Synthetic Aspirin-decursinol Adduct in Experimental Animal Models of Ischemic Stroke

نویسندگان

  • Bing Chun Yan
  • Joon Ha Park
  • Bich Na Shin
  • Ji Hyeon Ahn
  • In Hye Kim
  • Jae-Chul Lee
  • Ki-Yeon Yoo
  • In Koo Hwang
  • Jung Hoon Choi
  • Jeong Ho Park
  • Yun Lyul Lee
  • Hong-Won Suh
  • Jong-Gab Jun
  • Young-Guen Kwon
  • Young-Myeong Kim
  • Seung-Hae Kwon
  • Song Her
  • Jin Su Kim
  • Byung-Hwa Hyun
  • Chul-Kyu Kim
  • Jun Hwi Cho
  • Choong Hyun Lee
  • Moo-Ho Won
چکیده

Stroke is the second leading cause of death. Experimental animal models of cerebral ischemia are widely used for researching mechanisms of ischemic damage and developing new drugs for the prevention and treatment of stroke. The present study aimed to comparatively investigate neuroprotective effects of aspirin (ASA), decursinol (DA) and new synthetic aspirin-decursinol adduct (ASA-DA) against transient focal and global cerebral ischemic damage. We found that treatment with 20 mg/kg, not 10 mg/kg, ASA-DA protected against ischemia-induced neuronal death after transient focal and global ischemic damage, and its neuroprotective effect was much better than that of ASA or DA alone. In addition, 20 mg/kg ASA-DA treatment reduced the ischemia-induced gliosis and maintained antioxidants levels in the corresponding injury regions. In brief, ASA-DA, a new synthetic drug, dramatically protected neurons from ischemic damage, and neuroprotective effects of ASA-DA may be closely related to the attenuation of ischemia-induced gliosis and maintenance of antioxidants.

برای دانلود متن کامل این مقاله و بیش از 32 میلیون مقاله دیگر ابتدا ثبت نام کنید

ثبت نام

اگر عضو سایت هستید لطفا وارد حساب کاربری خود شوید

منابع مشابه

Protective Effect of Delayed Ischemic Postconditioning on Embolic Stroke Complications in Female Rat

Background & Aims: Ischemic postconditioning, conducted by a series of brief occlusion and release of the bilateral common carotid arteries, has neuroprotective properties in permanent or transient models of middle cerebral artery (MCA) occlusion but its delayed neuroprotective effects in the embolic model of stroke, especially in female rat, have not yet been reported and were investigated ...

متن کامل

The Neuroprotective Effect of Rosemary (Rosmarinus Officinalis L.) Hydroalcoholic Extract on Cerebral Ischemic Tolerance in Experimental Stroke

The prevention of BBB breakdown and the subsequent vasogenic edema are important parts of the medical management of ischemic stroke. The purpose of this study was to investigate the ischemic tolerance effect of Rosmarinus officinalis leaf hydro-alcoholic extract (RHE).Five groups of animals were designed: sham (underwent surgery without MCAO) and MCAO groups, the MCAO groups were pretreated ora...

متن کامل

P34: Berberin Exerts Neuroprotective Effects by Modulating Pro and Anti-Inflammatory Cytokines in Rat Model of MCAO

Many complicated mechanisms are involved in brain ischemia and the role of inflammatory factors in the progression of post-ischemic injury is inevitable. In present study, anti-inflammatory effect of berberine has been investigated in reperfusion injury after acute ischemic stroke. Male Wistar rats weighing 250-270 gr were randomly divided into four cohorts: healthy rats (control, n=20), sham-o...

متن کامل

The Neuroprotective Effect of Rosemary (Rosmarinus Officinalis L.) Hydroalcoholic Extract on Cerebral Ischemic Tolerance in Experimental Stroke

The prevention of BBB breakdown and the subsequent vasogenic edema are important parts of the medical management of ischemic stroke. The purpose of this study was to investigate the ischemic tolerance effect of Rosmarinus officinalis leaf hydro-alcoholic extract (RHE).Five groups of animals were designed: sham (underwent surgery without MCAO) and MCAO groups, the MCAO groups were pretreated ora...

متن کامل

The effect of pre-treatment with olive oil on TNFR1/NF-кB inflammatory pathway in rat ischemic stroke model

Introduction: Ischemic stroke is a serious neurological disease and a leading cause of death and severe disability in the world. A key component of the Mediterranean diet is olive oil, which contains compounds with antioxidant and anti-inflammatory effects. In this regard, the aim of the present study was to investigate the effect of olive oil on the ischemic damages and the inflammatory pathwa...

متن کامل

ذخیره در منابع من


  با ذخیره ی این منبع در منابع من، دسترسی به آن را برای استفاده های بعدی آسان تر کنید

برای دانلود متن کامل این مقاله و بیش از 32 میلیون مقاله دیگر ابتدا ثبت نام کنید

ثبت نام

اگر عضو سایت هستید لطفا وارد حساب کاربری خود شوید

عنوان ژورنال:

دوره 8  شماره 

صفحات  -

تاریخ انتشار 2013